BD-1047| CAS 138356-20-4

Cas No.:	138356-20-4
Chemical Name:	BD 1047 DIHYDROBROMIDE
Synonyms:	BD 1047 DIHYDROBROMIDE;N'-[2-(3,4-dichlorophenyl)ethyl]-N,N,N'-trimethylethane-1,2-diamine;N-[2-(3,4-DICHLOROPHENYL)ETHYL]-N-METHYL-2-(DIMETHYLAMINO)ETHYLAMINE DIHYDROBROMIDE;BD-1047;N-[2-(3,4-dichlorophenyl)ethyl]-N,N',N'-trimethylethane-1,2-diamine
SMILES:	CN(C)CCN(C)CCC1=CC(=C(C=C1)Cl)Cl
Formula:	C₁₃H₂₀N₂Cl₂
M.Wt:	275.2173
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

BD-1047 is a potent, selecitve Sigma 1 receptor (σ1) antagonist with Ki of 0.93 nM; displays 50-fold weaker affinity for sigma 2 receptor, and 100-fold selectivity over opiate, phencyclidine, muscarinic, dopamine, adrenoceptor and 5-HT receptors; attenuates the dystonia induced by DTG and haloperidol in rats.

MSDS

COA

LOT NO.	DOWNLOAD

2018-0101

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