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STD1T

  Cat. No.:  DC12503   Featured
Chemical Structure
893075-58-6
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More than 5000 active chemicals with high quality for research!
Field of application
STD1T (USP2a inhibitor STD1T) is a hit-to-lead, small-molecule inhibitor of USP2a with IC50 of 3.3 uM in Ub-AMC assays, displays no activity against USP7 at 10 uM.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 893075-58-6
Chemical Name: 2-(2-((5-(thiophen-2-yl)isoxazol-3-yl)methoxy)acetamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxamide
Synonyms: USP2a inhibitor STD1T
SMILES: C12CCCCC=1C(C(N)=O)=C(NC(=O)COCC1C=C(C3SC=CC=3)ON=1)S2
Formula: C19H19N3O4S2
M.Wt: 417.498
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Publication: 1. Tomala MD, et al. Eur J Med Chem. 2018 Apr 25;150:261-267.
Description: STD1T (USP2a inhibitor STD1T) is a hit-to-lead, small-molecule inhibitor of USP2a with IC50 of 3.3 uM in Ub-AMC assays, displays no activity against USP7 at 10 uM.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
2018-0101
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