DCC5029 |
Tap1a-opt1 |
Novel potent Na V -targeting peptide, exhibiting significant increased potency for Na V 1.1, Na V 1.2, Na V 1.3, Na V 1.6 and Na V 1.7 involved in several neurological disorders including acute and chronic pain, motor neuron disease and epilepsy |
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DCC5030 |
Tap1a-opt2 |
Novel potent Na V -targeting peptide, exhibiting significant increased potency for Na V 1.1, Na V 1.2, Na V 1.3, Na V 1.6 and Na V 1.7 involved in several neurological disorders including acute and chronic pain, motor neuron disease and epilepsy |
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DCC5031 |
Tapi-2 Acetate |
ADAM-17 (TACE) and MMP inhibitor, sensitizing cancer stem cells to the lethal effects of 5-FU and blocking shedding of TNF-α from cell membranes |
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DCC5032 |
Tariquidar Dimesylate |
Potent P-glycoprotein (P-gp) inhibitor |
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DCC5033 |
Tas-303 Hydrochloride |
Novel selective norepinephrine reuptake inhibitor, displaying significant norepinephrine transporter (NET) inhibitory activity toward the serotonin or dopamine transporters |
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DCC5034 |
tasidotin Hydrochloride |
Tubulin-binding dolastatin-15 analog, demostrating a wide spectrum of In Vivo antitumor activity |
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DCC5035 |
Tasp0233278 |
Potent and orally active V 1B receptor antagonist with antidepressant and anxiolytic activities in rodents |
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DCC5036 |
Tasp0277308 |
Potent and selective sphingosine 1-phosphate 1 (S1P1) receptor antagonist (IC50 = 7.8 nM) |
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DCC5037 |
Tasp0412098 |
Novel potent, selective, and orally active CRTH2 antagonist |
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DCC5038 |
Tat Peptide (47-57) |
Trans-activator of transcription (TAT) peptide, increasing Hepta-histidine (7H) permeability into cells for treatment of iPS cell-derived neurons carrying Tau or APP mutations suppressed Tau phosphorylation |
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DCC5039 |
Tat-gap19 |
Novel brain penetrant Cx43 hemichannel blocker |
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DCC5040 |
Tavarua Deoxyriboside A |
Potential neuroprotective agent, showing effects on cellular models of oxidative stress and neuroinflammation |
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DCC5041 |
Tazanolast |
Selective mast-cell-stabilizing agent, inhibiting ozone-induced airway hyperresponsiveness |
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DCC5042 |
Tb-2-081 |
Novel antagonist of IL-6 signaling |
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DCC5043 |
Tbbl-0000316 |
Novel antibiotic against Mycobacterium tuberculosis (Mtb), potently killing replicating, virulent Mtb H37Rv in a clavulanate-dependent manner |
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DCC5044 |
Tbdps-chc |
Novel potent MCT1 inhibitor, exhibiting good single agent anticancer efficacy properties |
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DCC5045 |
Tbe-31 |
Highly potent activator of Nrf2; Potent phase 2 cytoprotective pathway inducer and liver carcinogenesis blocker |
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DCC5046 |
Tbk1 Inhibitor-1 |
Novel TBK1/IKKε inhibitor |
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DCC5047 |
Tbz-07 |
Novel anti-angiogenesis and vascular disrupting agent, exhibiting moderate inhibitory cell proliferation activity |
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DCC5048 |
Tbz-19 |
Novel anti-angiogenesis and vascular disrupting agent, exhibiting moderate inhibitory cell proliferation activity |
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DCC5049 |
Tc299423 |
Novel agonist for nicotinic acetylcholine receptors (nAChRs), modestly selectively targeting α6β2 subtype |
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DCC5050 |
Tc-ac28 |
Novel potent and selective ligand of Brd2(2) |
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DCC5051 |
Tc-aqp1-1 |
Aquaporin 1 (AQP1) channel blocker |
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DCC5052 |
tc-c-14g |
Potent CB1 receptor inverse agonist |
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DCC5053 |
Tc-e 5006 |
Novel orally bioavailableγ-secretase modulator, reducing Aβ42 levels |
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DCC5054 |
FPR Agonist 43
Featured
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FPR Agonist 43 (compound 43) is a dual formyl peptide receptor 1 (FPR1) and formyl peptide receptor 2 (FPR2)/ALX agonist. |
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DCC5055 |
Tc-g1004 |
Potent and selective antagonist of adenosine A2A receptors |
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DCC5056 |
Tch-013 |
Non-competitive modulator of the proteasome inducing apoptosis a panel of myeloma and leukemia cell lines |
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DCC5057 |
Tc-i 2000
Featured
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Novel TRPM8 channel blocker |
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DCC5058 |
Tc-i 2014 |
Potent TRPM8 antagonist, exhibiting antiallodynic properties in pain models |
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