DCC0695 |
Ar-244555 |
Novel inverse agonist of Mas G-protein signaling, dose-dependently inhibiting inositol 1,4,5-trisphosphate accumulation in AdMas-infected cells, and attenuating the sarcomeric organization and cell enlargement observed in Mas overexpressing myocytes |
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DCC0696 |
Ar-a000002 |
Novel 5-hydroxytryptamine 1B (5-HT 1B ) autoreceptor antagonist |
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DCC0697 |
Ar-c117977 |
Novel immunosuppressant and monocarboxylate transporter inhibitor, reducing immune responses both in vitro and in vivo, maintaining long-term graft survival, and inducing operational tolerance |
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DCC0698 |
Ar-c141990 |
Novel inhibitor of lactate transporters (monocarboxylate transporters; MCTs) |
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DCC0699 |
Arc-1502 |
Highly potent CK2α inhibitor (K(i) = 0.5 nM), revealing high selectivity for CK2α in a panel of 140 protein kinases |
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DCC0700 |
Arc-3002 |
Highly potent and selective fluorescent probe of Rho kinase (ROCK) |
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DCC0701 |
Arcapillin |
Anticancer agent, inducing apoptosis mediated at least in part by the ERS pathway and inhibiting hepatoma tumor growth |
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DCC0702 |
Arcc-4nc |
Negative control for ARCC-4, binding androgen receptors (AR) without inducing degradation. |
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DCC0703 |
Arformoterol Hydrochloride |
Long-acting beta-2 adrenergic agonist |
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DCC0704 |
Arformoterol Maleate |
Long-acting beta-2 adrenergic agonist |
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DCC0705 |
Arg-arg-leu |
Potent tumor-homing tripeptide, targeting heat shock protein 70 (HSP70) |
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DCC0706 |
ari-3531 |
Novel selective inhibitor of PREP, displaying great selectivity over FAP, while also not inhibiting the DPPs. |
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DCC0707 |
arkin-1 |
Novel inhibitor of Ark1, the fission yeast member of the conserved Aurora kinase family |
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DCC0708 |
Arl-67085 |
P2T (P2YADP) purinoceptor antagonist |
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DCC0709 |
Arl-67156 |
Selective ecto-ATPase inhibitor, preventing metabolism of P2 purinoceptor agonists |
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DCC0710 |
Armeniaspirol A |
Natural inhibitor of recombinant purified ClpXP and ClpYQ AAA+ proteases, exhibitung potent antibacterial activity against H. pylori, including multidrug-resistant strains |
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DCC0711 |
Armillarisin A |
Regulator and promotor of immune functions, enhancing the role of macrophages, inhibiting bacteria growth, improving the protein metabolism, and regulating liver function |
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DCC0712 |
Arn2508 |
Novel dual inhibitor of the fatty acid amide hydrolase (FAAH) and the cyclooxygenase (COX) enzymes |
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DCC0713 |
Arn-810 Analog |
Novel selective estrogen receptor degrader (SERD), inducing regression in a tamoxifen-resistant breast cancer xenograft |
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DCC0714 |
Arq736 |
Novel potent and selective BRAF inhibitor |
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DCC0715 |
ar-r17779 |
Selective alpha-7 agonist |
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DCC0716 |
Arsai 1r |
The first human arylsulfatase A reversible inhibitor, impairing mouse oocyte fertilization |
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DCC0717 |
arvelexin |
Inhibitor of the inflammatory responses via NF |
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DCC0718 |
Arzoxifene Hydrochloride |
Non-steroidal selective estrogen receptor modulator (SERM) |
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DCC0719 |
As-0141 |
Novel Potent and Selective Inhibitor of CDC7 Kinase for the Treatment of Solid Cancers |
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DCC0720 |
As057278 |
Inhibitor of D-amino acid oxidase (DAAO) |
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DCC0721 |
As1069562 |
Inhibitor of serotonin (5-HT) and norepinephrine (NE) reuptake, significantly restoring decreased insulin-like growth factor 1 and fibroblast growth factor 2 mRNA levels in dorsal root ganglion and spinal cord, respectively |
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DCC0722 |
As1468240 |
Potent factor Xa inhibitor with significant oral anticoagulant activity |
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DCC0723 |
as1669058 |
Novel GPR119 agonist, potentiating insulin secretion from rat islets and having potent anti-diabetic effects in ICR and diabetic db/db mice |
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DCC0724 |
As1670542 |
Second-generation potent orally-active thrombopoietin (TPO) receptor agonist |
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