| Cat. No. | Product Name | Field of Application | Chemical Structure |
|---|---|---|---|
| DCC2437 | Gw305178x | Novel inhibitor of CDK |
|
| DCC2438 | Gw3333 | Novel selective and soluble inhibitor of tumor necrosis factor-alpha converting enzyme (TACE) |
|
| DCC2439 | gw409544 | Potent and selective full agonist for peroixisome proliferator-activated receptor-alpha |
|
| DCC2440 | Gw440139a | Novel potent RET kinase inhibitor |
|
| DCC2441 | gw441756 Hydrochloride | Potent TrkA kinase inhibitor |
|
| DCC2442 | Gw493838 | Novel agonist at the adenosine A1 receptor |
|
| DCC2443 | gw5638 | Orally active, nonsteroidal tamoxifen derivative and a ligand for the estrogen receptors (ERs), steroid receptor members of the nuclear receptor superfamily of transcription factors |
|
| DCC2444 | Gw568377a | Inhibitor of Mer Kinase, also inhibiting EGFR |
|
| DCC2445 | Gw612286x | Novel VEGFR inhibitor, also a moderate inhibitor of BET proteins with an IC 50 value of 4.6 μM for BRD4(1) |
|
| DCC2446 | Gw648495 | Potent inhibitor of PfDHODH, showing greater than 4,000-fold selectivity for the malarial enzyme |
|
| DCC2447 | gw693881a | Novel inhibitor of EGFR |
|
| DCC2448 | Gw701427a | Novel inhibitor of firefly luciferase derived from Photinus pyralis (FLuc), the most widely used luciferase |
|
| DCC2449 | Gw780056x | Selective cyclin dependent kinase inhibitor; Inhibitor of Yes1 kinase; Inhibitor of binding or entry into cells for Lassa Virus |
|
| DCC2450 | gw7845 | Selective agonist of peroxisome proliferator-activated receptor-γ (PPARγ) |
|
| DCC2451 | Gw807982x | Potent and selective inhibitor of glycogen synthase kinase 3 (GSK3) |
|
| DCC2452 | Gw809897x | Novel and potent inhibitor of VEGFR2 tyrosine kinase, non-selectivey inhibiting AURKA and AURKB |
|
| DCC2453 | Gw827106x | Potent GSK-3 inhibitor, highly selective over CDK-2 |
|
| DCC2454 | Gw833373x | Novel Inhibitor of GSK3beta |
|
| DCC2455 | Gw837016x | Novel inhibitor of mitosis and cytokinesis in T. brucei which causes human African trypanosomiasis (HAT) |
|
| DCC2456 | Gw844520 | Novel potent and selective inhibitor of the cytochrome bc1 complex of mitochondrial electron transport in P. falciparum |
|
| DCC2457 | gw853606 | Novel polo-like kinase (PLK1) inhibitor |
|
| DCC2458 | Gw856804x | Novel NAD+-competitive Sirt2 inhibitor |
|
| DCC2459 | Gwl-78 | Novel modulator of NF-Y transcription, inhibiting the binding of NF-Y to DNA, blocking cellular proliferation and cell cycle progression, interacting with a variety of CCAAT-containing promoters leading to p53-independent cell cycle arrest |
|
| DCC2460 | Gx-395 | Novel inhibitor of Nav1.7 |
|
| DCC2461 | Gx-585 | Novel potent inhibitor of NaV1.7 and highly selective against NaV1.5, having limited selectivity against NaV1.1 and NaV1.2 |
|
| DCC2462 | Gx-629 | GX-936 analog, antagonist of voltage-gated sodium 1.7 (Nav1.7) channels |
|
| DCC2463 | Gyki-53655 | AMPA antagonist |
|
| DCC2464 | Gyramide A | Novel bacterial DNA gyrase inhibitor, exhibiting antimicrobial activity and inhibiting bacterial cell division |
|
| DCC2465 | H-0104 Dihydrochloride | Novel Rho-associated coiled coil-formed protein kinase (ROCK) inhibitor, exerting strong intraocular pressure (IOP)-lowering effects into the eyes of monkeys |
|
| DCC2466 | H-0106 Dihydrochloride | Novel Rho-associated coiled coil-formed protein kinase (ROCK) inhibitor, exerting strong intraocular pressure (IOP)-lowering effects into the eyes of monkeys |
|
