DCC2947 |
kp1212 |
Novel non-chain terminating nucleoside analog anti-HIV inhibitor |
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DCC2948 |
Kpt-6604 |
Novel selective, orally bioavailable, PAK4 allosteric modulator against triple negative breast cancer |
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DCC2949 |
Kpu-300 |
Novel potent antimicrotubule agent, exhibiting potent cytotoxicity against HT-29 cells by strongly binding to tubulin and inducing microtubule depolymn. |
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DCC2950 |
Kr-12-a4 |
Potent antimicrobial peptide against gram-positive and gram-negative bacteria and relatively high LPS-neutralization activity |
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DCC2951 |
Kr-25210 |
Novel enteroviral replication inhibitor through a non-capsid binding mode with EC 50 values of 2.5, 2.2, and 3.7 μM against hRV B14, A21, and A71, respectively, targeting the replication stages in the virus |
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DCC2952 |
Kr-31762 |
Novel KATP channel opener, exerting cardioprotective effects by opening SarcKATP channels in rat models of ischemia/reperfusion-induced heart injury |
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DCC2953 |
Kras(g12c)-in-1 |
Novel irreversible inhibitor of KRAS(G12C) |
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DCC2954 |
Kras4b-in-d14 |
Novel specific inhibitor of oncogenic KRAS4b signaling, stabilizing the KRAS4b-PDEδ complex and remarkably decreasing tumor size and triggered apoptosis of tumor cells |
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DCC2955 |
Kras4b-pdeδ Stabilizer C19 |
Novel stabilizer of the KRAS4b-PDEδ complex, decreasing the proliferation of colorectal cancer cells, and increasing apoptosis via decreased activation of oncogenic KRAS4b signaling |
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DCC2956 |
Krc-108 |
Novel potent multi-kinase inhibitor, targeting Ron, Flt3 and TrkA as well as c-Met |
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DCC2957 |
Krc-327 |
Selective novel inhibitor of c-Met receptor tyrosine kinase with anticancer activity. |
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DCC2958 |
Krm-ii-08 |
Novel potent, non-toxic, blood-brain barrier crossing, α5-GABA A R preferring ligand, enhancing a chloride-anion efflux that induces mitochondrial membrane depolarization and in response, TP53 upregulation and p53, constitutively phosphorylated at S392, c |
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DCC2959 |
Krn4884 |
Potassium channel opener |
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DCC2960 |
Krn-8602 Hydrochloride |
Topo II inhibitor, exhibiting cytotoxic effects against tumour cells |
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DCC2961 |
Krp-109 |
Novel neutrophil elastase (NE) inhibitor, decreasing expression of TGF-ß Signal Related Genes |
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DCC2962 |
Krp-199 |
Highly potent and selective antagonist for the AMPA receptors, exhibiting good neuroprotective effects in vivo |
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DCC2963 |
Krp-204 |
Novel highly selective β3-adrenoceptor agonist being developed for the treatment of diabetes and obesity |
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DCC2964 |
Ks-133 |
Novel Potent and Selective VIPR2 Antagonist, Counteracting Cognitive Decline in a Mouse Model of Psychiatric Disorders |
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DCC2965 |
Ksc-392-150 |
Novel inhibitor of the permeability transition pore (PTP) |
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DCC2966 |
kscm-1 |
Selective ligand of the sigma-1 receptor |
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DCC2967 |
Kscm-11 |
Ligand of the sigma receptor |
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DCC2968 |
kscm-5 |
Ligand of the sigma receptor |
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DCC2969 |
Ksk120 |
Novel inhibitor of transcriptional activity in Chlamydia trachomatis |
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DCC2970 |
Ksl-128114 |
Novel, highly potent, and metabolically stable peptide inhibitor of syntenin, Inhibiting Glioblastoma |
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DCC2971 |
Kspa-1 |
Novel modulator of kinesin spindle protein (KSP)/Eg5, activating KSP-catalyzed ATP hydrolysis in the absence of microtubules yet inhibiting microtubule-stimulated ATP hydrolysis by KSP |
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DCC2972 |
Kt-182 |
Potent and selective inhibitor of ABHD6 |
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DCC2973 |
Kt2-962 |
TXA2/prostaglandin endoperoxide receptor antagonist |
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DCC2974 |
Kta-439 |
Thyroid hormone receptor β (TRβ) selective agonist |
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DCC2975 |
Ku-2285 |
Hypoxic cell radiosensitizer |
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DCC2976 |
Kufal194 |
Novel selective DYRK1A inhibitor |
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