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Retosiban

  Cat. No.:  DC41072  
Chemical Structure
820957-38-8
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More than 5000 active chemicals with high quality for research!
Field of application
Retosiban (GSK221149A) is a potent and selective oxytocin antagonist with a Ki of 0.65 nM.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 820957-38-8
Chemical Name: Retosiban
SMILES: O=C([C@@H](C1CC2=C(C=CC=C2)C1)N3)N([C@H](C4=COC(C)=N4)C(N5CCOCC5)=O)[C@H]([C@H](CC)C)C3=O
Formula: C27H34N4O5
M.Wt: 494.58
Sotrage: Please store the product under the recommended conditions in the Certificate of Analysis.
MSDS
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MSDS_24085_DC41072_820957-38-8
COA
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Cat. No. Product name Field of application
DC47258 Carbetocin acetate Carbetocin acetate, an oxytocin (OT) analogue, is an oxytocin receptor agonist with a Ki of 7.1 nM. Carbetocin acetate has high affinity to chimeric N-terminus (E1) of the oxytocin receptor (Ki=1.17 μM). Carbetocin acetate has the potential for postpartum hemorrhage research. Carbetocin acetate can crosse the blood-brain barrier and produces antidepressant-like activity via activation of oxytocin receptors in the CNS.
DC46970 L-372662 L-372662 is a potent and orally active non-peptide oxytocin antagonist with a Ki value of 4.8. The Kd value of L-372662 for wild-type hOTR and [A318G]OTR is 5.8 nM and 73 nM. L-372662 shows selectivity to OTR:V1aR.
DC45573 [Asp5]-Oxytocin [Asp5]-Oxytocin is the first 5-position neurohypophyseal hormone analogue possessing significant biological activity.
DC41072 Retosiban Retosiban (GSK221149A) is a potent and selective oxytocin antagonist with a Ki of 0.65 nM.
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