Novel Rho-associated coiled coil-formed protein kinase (ROCK) inhibitor, exerting strong intraocular pressure (IOP)-lowering effects into the eyes of monkeys

Novel full H1 agonist

Novel class of selective diacylglycerol acyltransferase 2 (DGAT2) inhibitor

Novel class of selective diacylglycerol acyltransferase 2 (DGAT2) inhibitor

Novel water-soluble and biocompatible small-molecule near-infrared II (NIR-II) fluorescent dye

Inhibitor of acetic acid-induced writhing response

Novel inhibitor of STAT3 activation, inhibiting head and neck cancer cell proliferation in a dose dependent manner

Inhibitor of monoamine oxidase (MAO)

Novel hemagglutinin (HA) protein inhibitor, inhibiting entry and replication of diverse influenza viruses via the HA protein, showing potent antiviral activity against diverse H1N1, H5N1, and H3N2 influenza viruses encoding HA proteins from both groups 1

Herbicide, being used for the control of broad-leaved weeds in cereals and oilseed rape

Topical corticosteroid with anti-inflammatory, antipruritic, and vasoconstrictor activities, inducing phospholipase A2 inhibitory proteins, activating gene expression of anti-inflammatory proteins mediated via the corticosteroid receptor response element

Antimalarial, binding to plasmpesin, a haemoglobin degrading enzyme unique to the malarial parasites

Selective peroxisome proliferator-activated receptor gamma (PPAR-gamma) modulator with antilipidemic activity

Novel HaloPROTAC degrader, inducing degradation of HaloTag fusion proteins

Novel Wnt inhibitor, blocking Wnt signaling downstream of beta-Catenin

Novel inhibitor of cathepsin K (CatK)

Novel selective inhibitor of Hap2/3/4/5p mediated transcription in vivo.

Natural antiproliferative, antifungal, antitumor agent, suppressing the epithelial-mesenchymal transition (EMT) process and inhibiting activation of the FAK/Src/STAT3 signaling pathway in A375 cells, targeting RACK1 to suppress cancer cell migration

Novel p300/CBP HAT inhibitor

Precursor for HATRIC-based ligand receptor capture (HATRIC-LRC)

Hepatocellular carcinoma (HCC)-selective cytotoxin, suppressing AKT anti-apoptotic signaling

Novel Inhibitor of Mycobacterium tuberculosis DosRST signaling and persistence