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Cat. No. Product name CAS No.
DC20407 HMPC

HMPC is a novel bacteriostatic agent that shows bacteriostatic activity against S. aureus (MIC=4 μg/ml) and rescues Caenorhabditis elegans from S. aureus infection.

128202-97-1
DC22107 HMS-101

HMS-101 (HMS101) is a potent, selective mutant IDH1 inhibitor, the IC50 is significantly lower in mouse bone marrow cells transduced with IDH1mut compared with IDH1wt (1 uM vs 12 uM, respectively).

1070690-06-0
DC9415 Hoechst 33342 (trihydrochloride)

Hoechst 33342 3Hcl(HOE 33342 3Hcl) is an AT-specific DNA minor groove ligand used fluorochrome for visualizing cellular DNA.

875756-97-1
DC9418 Hoechst 33258 analog

Hoechst stains are part of a family of blue fluorescent dyes used to stain DNA.

258843-62-8
DC22129 HOIPIN-1(JTP-0819958;HOIP inhibitor-1) Featured

HOIPIN-1 (JTP-0819958, HOIP inhibitor-1) is a chemical inhibitor of linear ubiquitin chain assembly complex (LUBAC, IC50=2.8 uM), specifically generates Met1-linked linear ubiquitin chains through the ubiquitin ligase activity in HOIP, and activates the N

DC22108 HOIPIN-8

HOIPIN-8 (HOIP inhibitor-8) is a potent chemical inhibitor of linear ubiquitin chain assembly complex (LUBAC, IC50=11 nM), specifically generates Met1-linked linear ubiquitin chains through the ubiquitin ligase activity in HOIP, and activates the NF-kB pa

DC10177 Homoplantaginin

Homoplantaginin is a flavonoid from a traditional Chinese medicine Salvia plebeia with antiinfammatory and antioxidant properties.

17680-84-1
DC12154 Hosenkoside A

Hosenkoside A is a baccharane glycoside isolated from the seeds of impatiens balsamina.

156791-82-1
DC12148 Hosenkoside B

Hosenkoside B is a baccharane glycoside isolated from the seeds of impatiens balsamina.

156764-82-8
DC12152 Hosenkoside F ((+)-Hosenkoside F)

Hosenkoside F is a baccharane glycoside isolated from the seeds of impatiens balsamina.

160896-45-7
DC12153 Hosenkoside K

Hosenkoside K is a baccharane glycoside isolated from the seeds of impatiens balsamina.

160896-49-1
DC12149 Hosenkoside M ((+)-Hosenkoside M)

Hosenkoside M is a baccharane glycoside isolated from the seeds of impatiens balsamina.

161016-51-9
DC23978 hPGDS-IN-1 Featured

hPGDS-IN-1 is a potent, selective hPGDS inhibitor with IC50 of 12 nM in FP or EIA assays..

1234708-04-3
DC23894 HPI-1 Featured

HPI-1 is a Hedgehog (Hh) pathway inhibitor that suppresses signaling through Shh (IC50=1.5 uM) without significantly affecting Wnt signaling (IC50>30 uM).

599150-20-6
DC12259 HS-10296 hydrochloride

HS-10296 hydrochloride is an orally available and third-Generation inhibitor of epidermal growth factor receptor (EGFR)-activating mutations and T790M-resistant mutation with limited activity against wild-type EGFR.

2134096-03-8
DC11128 HS148 Featured

HS148 (DAPK3 inhibitor HS148) is a selective DAPK3 inhibitor with Ki of 119 nM, >10-fold selectivity over Pim kinases..

1892595-16-2
DC12616 HS-152

HS-152 (HS152) is a specific small-molecule inhibitor of SMAD ubiquitin regulatory factor 1 (SMURF1), not only potently inhibits SMURF1-mediated RHOB degradation with IC50 of 3.2 uM, but also strongly blocks SMURF1-mediated RHOA and SMAD1 degradation (IC5

DC7426 HS-173 Featured

HS-173 is a potent PI3Kα inhibitor with IC50 of 0.8 nM.

1276110-06-5
DC12632 HS220 Featured

HS220 (HS-220) is a Plasmodium-selective takinib analog that targets atypical P. falciparum protein kinase 9 (PfPK9, Kd=4.1 uM) but does not inhibit HsTAK1, decreases K63-linked ubiquitination in P. falciparum; inhibits P. berghei parasite load in HuH7 ce

1570374-32-1
DC11126 HS56

HS56 (Pim-DAPK3 inhibitor HS56) is a potent, dual Pim/DAPK3 inhibitor with Ki of 72 nM (Pim-3) and 315 nM (DAPK3), shows micromolar potency toward Pim-1 and Pim-2 (Ki=1.5 and 17 uM).

922050-57-5
DC23784 HS-72

HS-72 is an allosteric, selective, cell-permeable inhibitor of inducible Hsp70 (Hsp70i or Hsp72), shows selectivity for Hsp70i over the closely related Hsc70 as well as the broader purinome.

1800285-51-1
DC21126 HSD 1169

HSD1169 is a potent, dual FLT3/TOPK inhibitor with activity against FLT3-ITD secondary mutations (D835 or F691, Kd=1-5 nM), potently inhibits acute myeloid leukemia cell lines (IC50=5 nM).

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