Cat. No. | Product name | CAS No. |
DC11528 |
Razuprotafib
Featured
Razuprotafib is a potent protein tyrosine phosphatase β (HPTPβ) inhibitor.. |
1008510-37-9 |
DC11549 |
Razuprotafib sodium
Razuprotafib sodium is a potent protein tyrosine phosphatase β(HPTPβ) inhibitor.. |
1809275-69-1 |
DC11161 |
RB-005
RB-005 (RB-005) is a potent, selective inhibitor of sphingosine kinase SphK1 (SK1) with IC50 of 3.6 uM, displays 15-fold selectivity over SphK2.. |
1425049-20-2 |
DC21558 |
RB-101
RB-101 is an mixed enkephalinase inhibitor that inhibits Aminopeptidase N and Neutral Endopeptidase with IC50 of 11 nM and 2 nM, respectively. |
135949-60-9 |
DC11430 |
RB-394
RB394 is an orally bioavailable and dual modulator of soluble epoxide hydrolase (sEH) and PPARγ. |
1830320-32-5 |
DC21559 |
RBPI-4
RBPI-4 is a selective small molecule inhibitor of poly(ADP-ribose) glycohydrolase (PARG) with IC50 of 3.0 uM, effectively inhibit PARG in cellular lysate.. |
1355339-07-9 |
DC12307 |
RCGD423
Featured
RCGD423 is a gp130 modulator, which prevents articular cartilage degeneration and promotes repair. |
108237-91-8 |
DC11135 |
RCM-1
RCM-1 (FOXM1 inhibitor RCM-1) is a nontoxic, small molecule that inhibits FOXM1 activity in vitro and in vivo, inhibits GFP-FOXM1 in U2OS cells with EC50 of 0.72 uM. |
339163-65-4 |
DC10993 |
RD162
RD162 is a second-generation, orally available antiandrogen that binds to androgen receptor (AR) with IC50 of 30.9 nM. |
915087-27-3 |
DC23821 |
REDX-05358
REDX-05358 is a novel potent, highly selective, orally bioavailable pan RAF inhibitor with IC50 of 0.1, 0.68, 0.171, and 0.076 nM for ARAF, BRAF, BRAF (V600E), and CRAF, respectively. |
1884226-20-3 |
DC22597 |
Regorafenib hydrochloride
Featured
Regorafenib hydrochloride (BAY73-4506) is a potent, orally active multikinase inhibitor that potently inhibits endothelial cell kinases in biochemical and cellular kinase phosphorylation assays with nanomolar range (IC50=3-200 nM). |
835621-07-3 |
DC21615 |
Relacatib
Relacatib (SB-462795, GSK-462795) is a potent and orally bioavailable small molecule cathepsin inhibitor with Ki of 41, 68 and 53 pM for cathepsin K, L and V, respectively. |
362505-84-8 |
DC20529 |
Remodelin Fluor
Remodelin Fluor is a small molecule analog of Remodelin, demonstrates in vivo activitiy against NAT10, significantly enhances the healthspan in a Lmna G609G HGPS mouse model.. |
1815580-35-8 |
DC8235 |
Repinotan (BAYx3702)
Repinotan is a high-affinity, selective, full agonist of the 5HT1A-receptor subtype with neuroprotective properties. |
144980-29-0 |
DC7261 |
Resminostat hydrochloride (4SC-201)
Resminostat(RAS2410; 4SC-201) is a potent inhibitor of HDAC1/3/6(IC50=43-72 nM); less potent to HDAC8 with IC50 of 877 nM. |
1187075-34-8 |
DC21561 |
BT-13
RET agonist BT13 is a novel small molecule GDNF receptor RET agonist, potently and selectively activates RET and its downstream intracellular signaling cascades in immortalized cells (EC50~20 uM). |
924537-98-4 |
DC4148 |
Retapamulin
Retapamulin is a topical antibiotic, which binds to both E. coli and S. aureus ribosomes with similar potencies with Kd of 3 nM. |
224452-66-8 |
DC20530 |
RET-IN-23c
RET-IN-23c is a potent and selective RET kinase inhibitor with IC50 of 61.2 nM, shows no significant inhibitory effect against VEGFR-2 and KDR. |
2095172-11-3 |
DC12234 |
Retinyl palmitate (Vitamin A palmitate; Retinol palmitate)
Retinyl palmitate is an ester of Retinol and is the major form of vitamin A found in the epidermis. Retinyl palmitate has been widely used in pharmaceutical and cosmetic formulations. |
79-81-2 |
DC23293 |
RETRA hydrobromide
RETRA hydrobromide is a small molecule mutant p53 reactivator that activates a set of p53-regulated genes and specifically suppresses mutant p53-bearing tumor cells in vitro and in mouse xenograft. |
1035875-01-4 |
DC23287 |
RETRA hydrochloride
RETRA hydrochloride is a small molecule mutant p53 reactivator that activates a set of p53-regulated genes and specifically suppresses mutant p53-bearing tumor cells in vitro and in mouse xenograft. |
1173023-52-3 |
DC23312 |
RETRA
RETRA is a small molecule mutant p53 reactivator that activates a set of p53-regulated genes and specifically suppresses mutant p53-bearing tumor cells in vitro and in mouse xenograft. |
1036069-26-7 |