DCC0845 |
Azd4619 |
Novel peroxisome proliferator-activated receptor alpha (PPARalpha) agonist, inducing alanine aminotransferase-1 gene and protein expression in human, but not in rat hepatocytes |
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DCC0846 |
Azd4996 |
Novel potent and highly selective cathepsin K inhibitor for the treatment of osteoarthritis |
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DCC0847 |
Azd5438-protac-8 |
First-in-class selective, partial CDK2 degrader against hearing loss and cancer, protecting against cisplatin ototoxicity and kainic acid excitotoxicity |
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DCC0848 |
Azd6370 |
Glucokinase activator, decreasing fasting and postprandial glucose in type 2 diabetes mellitus patients |
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DCC0849 |
Azd6564 |
Novel Fibrinolysis Inhibitor, Acting via Interference of a Protein-Protein Interaction |
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DCC0850 |
Azd6642 |
Novel selective inhibitor of 5-Lipoxygenase Activating Protein (FLAP) for the treatment of inflammatory diseases |
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DCC0851 |
Azd6703 |
Novel, potent and selective inhibitor of p38α MAP kinase |
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DCC0852 |
Azd7254 |
Novel potent smoothened inhibitor, demonstrating in vivo activity in abrogating the Hh paracrine pathway as well as anti- tumor effects |
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DCC0853 |
Azd9742 |
Antimicrobials, active against methicillin resistant S. aureus (MRSA) |
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DCC0854 |
Az-dyrk1b-33 |
Potent and selective ATP-competitive Dyrk1B kinase inhibitor |
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DCC0855 |
Azelastine |
Potent, second-generation, selective histamine-H1-receptor antagonist and mast cell stabilizer |
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DCC0856 |
Az-ghs-38 |
Novel CNS penetrant potent inverse agonist of GHS-R1a (IC 50 (affinity) = 0.77 nM) |
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DCC0857 |
Azide-a-dsbso
Featured
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Azide-A-DSBSO crosslinker is a mass spectrometry (MS)-cleavable, membrane-permeable, homobifunctional, azide-labeled, acid-cleavable cross-linked peptide. Azide-A-DSBSO crosslinker enables the study of protein-protein interactions via cross-linking mass spectrometry (XL-MS). |
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DCC0858 |
Azido-tpp1 |
Mitochondria-luciferin releasing agent, reacting with mitochondria-activatable luciferin (MAL-Probe), such as TPP-CL2, to release luciferin |
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DCC0859 |
Azithromycin Monohydrate |
Macrolide antibiotic, binding to the 50S subunit of the bacterial ribosome and thus inhibiting translation of mRNA |
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DCC0860 |
Azocholine |
Excellent photoswitchable agonist for neuronal α7 nAChRs |
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DCC0861 |
Azogw1929 |
Novel photoswitchable agonist for peroxisome proliferator-activated receptor γ (PPARγ) |
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DCC0862 |
Azolig 9 |
Novel photoswitchable ligand for the cannabinoid receptor 2 (CB2) |
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DCC0863 |
Azorosi-4 |
Novel photoswitchable agonist for peroxisome proliferator-activated receptor γ (PPARγ) |
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DCC0864 |
Az-pfkfb3-26 |
Potent and selective PFKFB3 inhibitor |
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DCC0865 |
Azumamide E |
Natural potent HDAC inhibitor |
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DCC0866 |
Az-vem |
Novel chimeric inhibitor of dimeric RAF, inhibiting B-Raf V600E mutan |
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DCC0867 |
B07 Hydrochloride |
Novel CCR5 antagonist-based HIV-1 entry inhibitor |
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DCC0868 |
Ba-53038b |
Novel HBV core protein allosteric modulator (CpAM), bing to the HAP pocket and modulating HBV capsid assembly in a distinct manner |
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DCC0869 |
Baa485 |
Novel activator of Pyrin inflammasome |
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DCC0870 |
Bace1-in-cpd C |
Novel potent nonbrain-penetrant BACE1 inhibitor |
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DCC0871 |
Baclmk |
Allosteric Inhibitor of the NS2B-NS3 Protease from Dengue Virus |
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DCC0872 |
Bag-1 Inhibitor Thio-2 |
Novel inhibitor of BAG-1-mediated protein interactions, targeting the RAF-MEK-ERK signaling pathway, transformed cells |
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DCC0873 |
Bak2-66 |
Selective Dopamine D3 Receptor Antagonist |
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DCC0874 |
Bal101553 Dihydrochloride |
Novel microtubule inhibitor as the prodrug of BAL27862, activating spindle assembly checkpoint, exerting antiproliferative effects and dose-dependent vascular disruption |
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