DCC2269 |
Gls1 Inhibitor Ll202 |
Novel inhibitor of glutaminase 1 (GLS1) with high binding affinity (SPR, Kd = 24 nM; ITC, Kd = 37 nM), exhibiting a similar in vivo antitumor activity as CB839 |
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DCC2270 |
Glut4-activator-26b |
Novel potent glucose transporter type 4 (GLUT4) translocation activator, showing a significant blood glucose lowering effect in the severe diabetic mice model |
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DCC2271 |
Glut-i1 |
Selective inhibitor of human glucose transporter subtype 1/4 (hGLUT1/4) |
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DCC2272 |
Glut-i2 |
Selective inhibitor of human glucose transporter subtype 1/4 (hGLUT1/4) |
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DCC2273 |
Glut-i2-nh2 |
Glucose transporter inhibitor linker for insulin conjugate |
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DCC2274 |
Glut-in-30 |
Novel glucose transporter (GLUT) inhibitor, exhibited high antitumor potency through the suppression of glucose uptake (IC 50 : 2.5 μM), while not cytotoxic to prostate and mammary epithelial cells |
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DCC2275 |
Glycitin 6"-o-malonate |
Metabolite of soy isoflavones, promoting the proliferation of bone marrow stromal cells and osteoblasts and suppresses bone turnover |
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DCC2276 |
Gm3 N-12 |
Novel GM3 derivative, showing excellent migration and invasion inhibitory effects in cells and marked antitumor activity in C57BL/6 mice, involving focal adhesion and ECM-receptor interaction signaling pathways |
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DCC2277 |
Gma-839 |
Selective modulator of gamma-aminobutyric acid(A) receptors |
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DCC2278 |
Gmb-805 |
Novel potent BCR-Abl PROTAC, inducing degradation and demonstrating in vivo activity |
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DCC2279 |
Gmb-905 |
Negative control for GMB-805 |
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DCC2280 |
Gn39482 |
Novel Tubulin Polymerization Inhibitor |
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DCC2281 |
Gne-0723 |
Novel GluN2A subunit-selective and brain-penetrant positive allosteric modulator (PAM) of The N-methyl-d-aspartate receptor (NMDAR) |
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DCC2282 |
Gne-0946 |
Novel potent and selective RORc inverse agonist |
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DCC2283 |
Gne-203 |
Novel Met inhibitor |
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DCC2284 |
Gne-3476 |
Novel GluN2A-selective NMDA receptor positive allosteric modulator (PAM) |
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DCC2285 |
Gne-5729 |
Novel NMDAR PAM with both an improved pharmacokinetic profile and increased selectivity against AMPARs |
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DCC2286 |
Gne-618 |
Novel inhibitor of nicotinamide phosphoribosyl transferase (NAMPT) |
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DCC2287 |
Gne-6689 |
Negative control for GNE-2256 |
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DCC2288 |
Gne-6901 |
Novel GluN2A-selective NMDA receptor positive allosteric modulator (PAM) |
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DCC2289 |
Gne-783 |
Novel selective CHK1 inhibitor |
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DCC2290 |
Gnf351 |
Novel potent aryl hydrocarbon receptor (AHR) antagonist with the capacity to inhibit both DRE-dependent and -independent activity |
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DCC2292 |
Gnf-pf-3539 |
Novel Inhibitor of EGF-EGFR Interactions |
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DCC2293 |
Gnf-pf-3600 |
Novel inhibitor of Plasmodium falciparum, killing both blood- and sexual-stage P. falciparum parasites |
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DCC2294 |
gnf-pf-3834 |
Dose dependent up-regulator of the level of E-cadherin in SW620 cells |
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DCC2295 |
Gnidimacrin |
Natural highly potent HIV latency-reversing agent |
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DCC2296 |
Gnlpt-in-1 |
Novel inhibitor of Gram-negative lipoprotein trafficking |
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DCC2297 |
Gnmt Inducer K-117 |
Novel potent GNMT inducer, inhibiting Huh7 cell growth in vitro and xenograft in vivo |
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DCC2298 |
Go/ldha-in-7 |
Dual Glycolate Oxidase/Lactate Dehydrogenase A (GO/LDHA) Inhibitor for Primary Hyperoxaluria |
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DCC2299 |
Gonadorelin Acetate |
Agonist of the GnRH receptor, inducing the secretion of the gonadotropins follicle-stimulating hormone and luteinizing hormone from the pituitary gland and to increase sex hormone production by the gonads |
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