DCC2225 |
Gc-204 |
Selective inhibitor of carbonic anhydrase IX (CAIX) |
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DCC2226 |
Gc-205 |
Selective inhibitor of carbonic anhydrase IX (CAIX) |
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DCC2227 |
Gca-186 |
Highly potent non-nucleoside inhibitor of HIV-1 reverse transcriptase |
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DCC2228 |
Gcc5694a |
Novel Potent and Selective Sodium Glucose Co-Transporter 2 (SGLT2) Inhibitor for the Treatment of Type 2 Diabetes |
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DCC2229 |
Gcs Inhibitor Bz1 |
Novel glucosylceramide synthase (GCS) inhibitor, rescuing lysosomal deficits, α-synuclein pathology and neuron toxicity |
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DCC2230 |
Gdc0575 |
Novel highly-selective oral checkpoint kinase 1 (Chk1) inhibitor |
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DCC2231 |
Gdc-0575 Dihydrochloride |
Novel potent, selective and orally bioavailable Chk1 inhibitor |
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DCC2232 |
Gdc-0834 |
Novel Bruton's tyrosine kinase (BTK) inhibitor |
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DCC2233 |
Gdc-0917 |
Novel SMAC mimetic and IAP antagonist |
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DCC2235 |
Gdk-100017 |
Inhibitor of the Wnt/beta-catenin signaling pathway, suppressing cell proliferation and enhancing radiosensitivity in A549/Wnt2 cells. |
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DCC2236 |
Gebr-7b |
Novel Phosphodiesterase 4D (PDE4D) Inhibitor |
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DCC2237 |
Geiparvarin |
MAO inhibitor |
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DCC2238 |
Genaconazole |
Novel antifungal agent |
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DCC2239 |
Geneseroline |
Metabolite of ganstigmine, a novel acetylcholinesterase inhibitor |
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DCC2240 |
Geopyxin C |
Natural covalent Cys151-dependent NRF2 activator |
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DCC2241 |
Geopyxin F |
Natural non-covalent NRF2 activator, activating NRF2 in A KEAP1-dependent but Cys151-independent manner, conferring greater protection than a Cys151-dependent analog, geopyxin C |
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DCC2242 |
GFB-12811
Featured
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GFB-12811 is a high selective and orally active CDK5 inhibitor with an IC50 of 2.3 nM. GFB-12811 is highly selective over the other tested kinases (CDK1/2/6/7/9). |
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DCC2243 |
G-glu-glu |
Endogenous dipeptide, activating N-methyl-D-aspartate receptors |
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DCC2244 |
Ghsr Inverse Agonist 29 |
Novel nonpeptidic inverse agonist of the Ghrelin Receptor (GHSR) |
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DCC2245 |
Gi-129471 |
Metalloproteinase inhibitor, specifically blocking TNF-alpha secretion both in vitro and in vivo |
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DCC2246 |
Gi261520a |
Potent EGFR/erbB2 dual inhibitor |
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DCC2247 |
Gic-1001 |
Novel oral anti-nociceptive agent, showing peripheral opioid agonistic activity and hydrogen sulphide-releasing capacity |
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DCC2248 |
Gidazepam |
Potent mitochondrial benzodiazepine receptors (MBRs) ligand; Prodrug for its active metabolite bromo-nordazepam |
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DCC2249 |
Gif-0854-r |
Novel suppressor of endoplasmic reticulum (ER) stress and oxidative stress, preventing protein aggregate accumulation in vitro and in cultured hippocampal HT22 neuronal cells, as well as glutamate-induced oxytosis and erastin-induced ferroptosis |
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DCC2250 |
Gif-0856-r |
Novel suppressor of endoplasmic reticulum (ER) stress and oxidative stress, preventing protein aggregate accumulation in vitro and in cultured hippocampal HT22 neuronal cells, as well as glutamate-induced oxytosis and erastin-induced ferroptosis |
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DCC2251 |
Gilteritinib Fumarate
Featured
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Gilteritinib (ASP2215) hemifumarate is a potent and ATP-competitive FLT3/AXL inhibitor with IC50 of 0.29 nM/0.73 nM, respectively. |
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DCC2252 |
Ginkgonitroside |
Natural suppressor of mesenchymal stem cell (MSC) differentiation |
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DCC2253 |
Ginnalin A |
Natural Activator of the Nrf2-Regulated Antioxidant Defense System in SH-SY5Y Cells, Binding to the Subpockets of Keap1 Kelch Domain |
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DCC2254 |
Gk-136901 |
First-in-Class, Potent, and Orally Bioavailable NADPH Oxidase Isoform 4 (Nox4) Inhibitor |
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DCC2255 |
Gk-667 |
Novel water solubile prodrug of ICRF-193, penetrating into NVCMs, reaching intracellular concentrations sufficient to induce cytoprotective effects against ANT toxicity |
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