DCC2256 |
Gka-22 |
Novel Allosteric Activator of Human Glucokinase in the Absence of Glucose |
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DCC2257 |
Gka-71 |
Novel and potent glucokinase activator (GKA) |
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DCC2258 |
Gkm001 |
First-in-class liver-selective glucokinase activator for the treatment of type 2 diabetes |
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DCC2259 |
glaziovianin A |
Novel inhibitor of the cell cycle progression in M-phase; Inhibotor of endosome maturation |
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DCC2260 |
Glenvastatin |
Novel 3-hydroxy-3-methylglutaryl coenzyme A reductase inhibitor |
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DCC2261 |
Glft2-in-31 |
Novel Galactofuranosyltransferase 2 (GlfT2) inhibitor |
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DCC2262 |
Glipentide |
Second-generation sulfonylurea, promoting the accumulation of fructose 2,6-bisphosphate in hepatocytes |
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DCC2263 |
Glmu-in-5175178 |
Novel inhibitor of the acetyltransferase activity of Escherichia coli N-acetylglucosamine-1-phosphate-uridyltransferase/glucosamine-1-phosphate-acetyltransferase (GlmU). |
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DCC2264 |
Glo1-in-60 |
Novel potent Glyoxalase 1 (GLO1) inhibitor, demonstrating to penetrate the blood-brain barrier, elevating levels of methylglyoxal in the brain, and reducing depression-like behavior in mice |
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DCC2265 |
Glo1-in-9 |
Novel inhibitor of glyoxalase 1 (Glo1), increasing the cellular methylglyoxal levels in human cells and suppressing the osteoclast formation of mouse bone marrow-derived macrophages |
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DCC2266 |
Glp-2 (1-33) Acetate |
Enteroendocrine hormone, stimulating the growth of intestinal epithelium |
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DCC2267 |
Glp-2r Modulator I |
Ago-allosteric modulator of human GLP-2R |
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DCC2268 |
Glpg0259 |
The first-in-class, ATP-competitive inhibitor of MAPKAPK5 |
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DCC2269 |
Gls1 Inhibitor Ll202 |
Novel inhibitor of glutaminase 1 (GLS1) with high binding affinity (SPR, Kd = 24 nM; ITC, Kd = 37 nM), exhibiting a similar in vivo antitumor activity as CB839 |
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DCC2270 |
Glut4-activator-26b |
Novel potent glucose transporter type 4 (GLUT4) translocation activator, showing a significant blood glucose lowering effect in the severe diabetic mice model |
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DCC2271 |
Glut-i1 |
Selective inhibitor of human glucose transporter subtype 1/4 (hGLUT1/4) |
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DCC2272 |
Glut-i2 |
Selective inhibitor of human glucose transporter subtype 1/4 (hGLUT1/4) |
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DCC2273 |
Glut-i2-nh2 |
Glucose transporter inhibitor linker for insulin conjugate |
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DCC2274 |
Glut-in-30 |
Novel glucose transporter (GLUT) inhibitor, exhibited high antitumor potency through the suppression of glucose uptake (IC 50 : 2.5 μM), while not cytotoxic to prostate and mammary epithelial cells |
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DCC2275 |
Glycitin 6"-o-malonate |
Metabolite of soy isoflavones, promoting the proliferation of bone marrow stromal cells and osteoblasts and suppresses bone turnover |
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DCC2276 |
Gm3 N-12 |
Novel GM3 derivative, showing excellent migration and invasion inhibitory effects in cells and marked antitumor activity in C57BL/6 mice, involving focal adhesion and ECM-receptor interaction signaling pathways |
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DCC2277 |
Gma-839 |
Selective modulator of gamma-aminobutyric acid(A) receptors |
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DCC2278 |
Gmb-805 |
Novel potent BCR-Abl PROTAC, inducing degradation and demonstrating in vivo activity |
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DCC2279 |
Gmb-905 |
Negative control for GMB-805 |
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DCC2280 |
Gn39482 |
Novel Tubulin Polymerization Inhibitor |
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DCC2281 |
Gne-0723 |
Novel GluN2A subunit-selective and brain-penetrant positive allosteric modulator (PAM) of The N-methyl-d-aspartate receptor (NMDAR) |
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DCC2282 |
Gne-0946 |
Novel potent and selective RORc inverse agonist |
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DCC2283 |
Gne-203 |
Novel Met inhibitor |
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DCC2284 |
Gne-3476 |
Novel GluN2A-selective NMDA receptor positive allosteric modulator (PAM) |
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DCC2285 |
Gne-5729 |
Novel NMDAR PAM with both an improved pharmacokinetic profile and increased selectivity against AMPARs |
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