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Upidosin

  Cat. No.:  DC72329   Featured
Chemical Structure
152735-23-4
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More than 5000 active chemicals with high quality for research!
Field of application
Upidosin (Rec 15/2739) is an α-1 adrenoceptor (α-1 AR) antagonist. Upidosin shows moderate selectivity for the α-1A AR subtype. Upidosin shows uroselectivity in urethra and prostate with a Kb value of 2-3 nM higher than in ear artery and aorta with a Kb value of 20-100 nM. Upidosin inhibits [3H]prazosin binding to cloned human α-1A adrenergic receptor. Upidosin can be used for the research of urethral obstruction.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 152735-23-4
Chemical Name: 4H-1-Benzopyran-8-carboxamide,N-[3-[4-(2-methoxyphenyl)-1-piperazinyl]propyl]-3-methyl-4-oxo-2-phenyl-
Synonyms: 4H-1-Benzopyran-8-carboxamide,N-[3-[4-(2-methoxyphenyl)-1-piperazinyl]propyl]-3-methyl-4-oxo-2-phenyl-;N-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]-3-methyl-4-oxo-2-phenylchromene-8-carboxamide;AC1L3XX2;ACMC-20n6iu;Rec 15-2739;Rec-15-2739;SB 216469-S;UNII-TXG28R7G4Y;UPIDOSIN;L000508;Q27089098;TXG28R7G4Y;SB 216469;NS00121149;CS-0026991;N-(3-(4-(o-Methoxyphenyl)-1-piperazinyl)propyl)-3-methyl-4-oxo-2-phenyl-4H-1-benzopyran-8-carboxamide;Upidosin [INN];Rec 15/2739;GTPL496;CHEMBL278865;SB 216469 BASE;HY-106954;DTXSID70165115;Rec 15/2739; Recordati 15/2739; SB 216469;MS-29497;152735-23-4;SB-216469;AKOS030553705;4H-1-Benzopyran-8-carboxamide, N-(3-(4-(2-methoxyphenyl)-1-piperazinyl)propyl)-3-methyl-4-oxo-2-phenyl-;BDBM50057465;3-Methyl-4-oxo-2-phenyl-4H-chromene-8-carboxylic acid {3-[4-(2-methoxy-phenyl)-piperazin-1-yl]-propyl}-amide;SCHEMBL6638869;N-(3-(4-(2-nethoxyphenyl)-1-piperazinyl)propyl)-3-methyl-4-oxo-2-phenyl-4H-1-benzopyran-8-carboxamide monomethane sulfonate monohydrate;DA-68488;DA-68488
SMILES: COC1C=CC=CC=1N1CCN(CCCNC(C2C3=C(C(=O)C(C)=C(C4C=CC=CC=4)O3)C=CC=2)=O)CC1
Formula: C31H33N3O4
M.Wt: 511.61142
Purity: 98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
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MSDS_36780_DC72329_152735-23-4
COA
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Cat. No. Product name Field of application
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