DCC0276 |
5-cltep |
HIV-1 integrase inhibitor |
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DCC0277 |
5-formylcytosine |
Rare base found in mammalian DNA, having functional roles in DNA that go beyond being a demethylation intermediate |
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DCC0278 |
5-fu Prodrug 4 |
Novel palladium-activated 5-FU prodrug, being completely innocuous to cells and highly resistant to metabolization by primary hepatocytes and liver S9 fractions (the main metabolic route for 5-FU degradation), and rapidly converted into 5-FU in the presen |
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DCC0279 |
5-hiaa |
Serotonin metabolite, systemically inhibiting RAS/MAPK signaling in different organs of C. elegans |
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DCC0280 |
5-ht2c Agonist 58 |
Novel selective 5-HT 2C agonist with >300-fold functional selectivity over 5-HT 2B and >70-fold functional selectivity over 5-HT 2A , reducing food intake in an acute rat feeding model |
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DCC0281 |
5-ht3 Antagonist-4i
Featured
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5-HT3 antagonist 4 is a 5-HT3 receptor (5HT3R) antagonist. 5-HT3 antagonist 4 prevents diabetes-induced depressive phenotypes in mice. |
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DCC0282 |
5-ht7r Antagonist 2c |
Novel potent and selective G protein-biased 5-HT 7 R Antagonist, significantly reducing self-grooming duration time to the level of wild-type mice |
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DCC0283 |
5-hydroxydantrolene |
Metabolite of dantrolene |
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DCC0284 |
5'-hydroxydatiscetin |
Morin isomer, antioxidant |
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DCC0285 |
5-hydroxydiclofenac |
Active metabolite of diclofenac, targeting COX and CaMKIIα hub domain |
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DCC0286 |
5-mca-nat |
Melatonin analogue, selectively binding on MT3 subsites |
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DCC0287 |
5-methoxyleoligin |
Natural proangiogenic agent, downregulating the cellular uptake of all- trans-retinoic acid (atRA) under hypoxia |
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DCC0288 |
5-methyl-ds2 |
Novel potent δ-selective allosteric modulator, displayed at least 60-fold selectivity for α4β1δ over α4β1γ2 receptor subtypes, Ki(α4β1δ |
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DCC0289 |
5-mpep |
Neutral allosteric site ligand of the metabotropic glutamate receptor subtype 5 (mGlu5), blocking the effects of both the allosteric antagonist MPEP and potentiator CDPPB |
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DCC0290 |
5n-bicalutamide |
Novel highly potent nonsteroidal antiandrogen (NSAA) |
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DCC0291 |
5-oh-hxmf |
Inducer of neurite outgrowth via cAMP/PKA/CREB pathway in PC12 cells |
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DCC0292 |
5-oh-phip |
PhIP metabolite |
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DCC0293 |
5'-o-methyl-3-hydroxyflemingin A |
Natural inhibitor of hedgehog (Hh) signal transduction, diminishing characteristics of cancer stem cells, leading to decreasing production of the Hh target proteins BCL2, PTCH1, and BMI1 |
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DCC0294 |
5'-o-tritylthymidine |
Blocker of the formation of the FAK/Mdm-2 complex; subsequently, activating p53 and caspase-8 and leading to increase detachment and apoptosis in breast and colon cancers |
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DCC0295 |
5sglcnhex |
Novel O-GlcNAc transferase (OGT) inhibitor, inducing dose- and time-dependent decreases in O-GlcNAc levels |
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DCC0296 |
5'-ß-l-asp-fudr |
Novel FUdR prodrug. possessing a better tumor inhibition rate and a better metabolic stability than FUdR through a ATB0, -mediated prodrug approach |
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DCC0297 |
6"-o-acetyldaidzin |
Metabolite of soy isoflavone; Antioxidant |
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DCC0298 |
6"-o-acetylgenistin |
Metabolite of soy isoflavones |
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DCC0299 |
6"-o-malonyldaidzin |
Metabolite of soy isoflavones |
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DCC0300 |
6,6''-biapigenin |
Potent and selective nociceptin opioid receptor (NOP) agonist |
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DCC0301 |
6,7,3',4'-tetrahydroxyflavone |
Novel potent MtbCoaBC inhibitor (IC50: 0.08 µM) |
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DCC0302 |
6,8-diprenyleriodictyol |
Antioxidant, inhibiting Cu(2+)-mediated oxidation of human low density lipoprotein (LDL) |
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DCC0303 |
65-a11 |
Novel methuselah (Mth)-specific antagonist |
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DCC0304 |
680sir |
Novel fluorescent probe for near-IR live-cell super-resolution imaging |
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DCC0305 |
6-alkynyl-fucose |
Widely used fucosylation probe, strongly inhibiting fucosylation and GDP-fucose synthetase FX, halting hepatoma invasion |
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