Bis-propargyl-PEG9 is a crosslinker containing two propargyl groups at each terminal end. The propargyl groups can be reacted with azide-bearing compounds or biomolecules via copper catalyzed azide-alkyne Click Chemistry to yield stable triazole linkages.

Propargyl-PEG4-amine is a PEG derivative containing a propargyl group and an amine group. The amine group is reactive with carboxylic acids, activated NHS esters, carbonyls (ketone, aldehyde) etc. The propargyl group can be reacted with azide-bearing compounds or biomolecules via copper catalyzed azide-alkyne Click Chemistry to yield a stable triazole linkage. PEG Linkers can be useful in the development of antibody drug conjugates (ADCs).

Sulfo-SANPAH Crosslinker, or N-Sulfosuccinimidyl-6-[4'-azido-2'-nitrophenylamino] hexanoate is a water soluble, heterobifunctional protein crosslinker with a spacer arm length of 18.2 angstroms.

ACS67 is an F-series prostaglandin (PG) analog for treatment of glaucoma. ACS 67 reduces intra-ocular pressure (IOP) and increases levels of reduced glutathione and cGMP in the aqueous humor of glaucomatous pigmented rabbits. ACS67 also acts as a neuroprotectant that stimulates GSH levels.

Halosulfuron-methyl is a common herbicide.

Pirenoxine, also known as Catalin, is an anti-cataractogenesis agent which interacts with selenite or calcium ions that have been proven as factors leading to the formation of lens cataract.

3-Cl-DPA is an activator of cardiac troponin by a mechanism distinct from bepridil or TFP.

DCAI hydrochloride is an inhibitor of nucleotide exchange and nucleotide release, by binding to the pocket adjacent to the Ras-SOS interface.

STAT3-IN-8 is a cell permeable JAK1/JAK2/TYK2/STAT3 activation inhibitor.

Oxathiapiprolin is a oomycete fungicide, targeting an oxysterol binding protein.

Englerin A is a natural potent activator of ion channels formed by Transient Receptor Potential Canonical 4 and 5 proteins (TRPC4 and TRPC5).

TFIIH Modulator-12 is a small molecule destabilization inducer of the trichothiodystrophy group A protein (TTD-A or p8) dimerization which modulates TFIIH transcriptional activity.

NHNB is a selective inhibitor of histone deacetylases-8 (HDAC8). NHNB provides the most potent CE4 inhibitor reported to date.

Nothofagin is a natural anti-oxidant which inhibits endothelial protein C receptor (EPCR) shedding. Nothofagin shows diuretic, natriuretic, and potassium-sparing effects associated with prostanoids generation and muscarinic receptor activation.

Lumiflavine is a riboflavin uptake inhibitor. Lumiflavine is produced by the photolysis of vitamin B2 (Riboflavin).

Epigenetic Multiple Ligand is a cell-permeable inhibitor of substrate processing by several chromatin-associated enzymes, including SIRT1/2, H3/SET7, H3/p300/CBP, H4/RmtA, PABP1/CARM1, and H4/PRMT1. It acts by inducing either apoptosis or granulocytic differentiation.

AC-93253 iodide is a SIRT2 selective inhibitor. It acts by significantly enhancing acetylation of tubulin, p53, and histone H4.

CAY10589 is an inhibitor of mPGES-1.

MK6-83 is an agonist of the transient receptor potential channel ML3 (TRPML3).

TT01001 is a mitoNEET ligand. It acts by improving diabetes and ameliorates mitochondrial function in db/db mice.

KS370G is an inhibitor of UUO-induced renal fibrosis markers expression. It acts by attenuating collagen deposition in the obstructed kidney and significantly lowering the expression of renal inflammatory chemokines/adhesion molecules and monocyte cells marker.

S32826 is an inhibitor of autotaxin.

5HPP-33 is an antiproliferative and antimitotic microtubule-stabilizer.

Atractyloside Potassium Salt is a natural inhibitor of ADP and ATP transport (AAT). It acts by binding specifically to the adenine nucleotide translocator in the inner mitochondrial membrane.

Barnidipine Hydrochloride is a long-acting calcium channel blocker.

CAPE is an inhibitor of BAF. It works by activating latent HIV-1, inhibiting PDGF-induced proliferation of vascular smooth muscle cells through the activation of p38 mitogen-activated protein kinase (MAPK), hypoxia-inducible factor (HIF)-1alpha and subsequent induction of heme oxygenase-1 (HO-1).

5-Methyltryptamine hydrochloride acts as a 5-HT receptor agonist.

Hyodeoxycholic acid sodium salt is a natural secondary bile acid. It improves high-density lipoprotein (HDL) function, reduces farnesoid X receptor antagonist bile acids and the gene expression levels of sterol regulatory element binding protein 1c, acetyl-CoA carboxylase, fatty acid synthase, and stearoyl-CoA desaturase-1, and induces strong cytotoxicity, apoptosis and IL-8 synthesis.

Lomifylline is an inducer of Ca2±release from intracellular stores via the ryanodine receptor.

Temafloxacin is an antibiotic and antimycobacterial agent. It was approved to treat lower respiratory tract infections, genital and urinary infections like prostatitis, and skin infections in 1992.