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Cat. No. Product Name Field of Application Chemical Structure
DCAPI1014 Eplerenone Featured Eplerenone, also known as Inspra and CGP-30083, is a selective aldosterone receptor antagonist used to treat hypertension and congestive heart failure. Eplerenone provides marked protection against vascular injury in the kidney and heart.
DC23786 Epolactaene Epolactaene is a neuritogenic fungal isolate that arrests the cell cycle at the G0/G1 phase and induces the outgrowth of neurites in human neuroblastoma SH-SY5Y cells.
DC7120 Epothilone A Epothilone A is a Taxol-like microtubule-stabilizing agent that induces tubulin polymerization, leading to cell cycle arrest at the G2-M transition, cytotoxicity, and apoptosis.
DC4198 Epothilone B Featured Epothilone B is a Taxol-like microtubule-stabilizing agent with EC0.01 of 1.8 μM.
DC7012 Epothilone D Epothilone D(Desoxyepothilone B; KOS 862) is a natural polyketide compound isolated from the myxobacterium Sorangium cellulosum.
DC8030 Epoxomicin Featured Epoxomicin is a selective and irreversible inhibitor of 20S proteasome with an IC50 value of 4 nM.
DC12311 Eprobemide (LIS 630) Featured Eprobemide is a non-competitive reversible inhibitor of monoamine oxidase A.
DC9171 Eprosartan mesylate Eprosartan is a nonpeptide angiotensin II receptor antagonist with IC50 of 9.2 and 3.9 nM in rat and human adrenal cortical membranes, respectively.
DC9260 Eptapirone Featured Eptapirone (F-11,440) is a very potent and highly selective 5-HT1A receptor full agonist of the azapirone family.
DC5182 EPZ004777 Featured EPZ004777 is a potent, selective DOT1L inhibitor with IC50 of 0.4 nM.
DC7121 EPZ005687 Featured EPZ-005687 is a potent and selective inhibitor of EZH2 with Ki of 24 nM, 50-fold selectivity against EZH1 and 500-fold selectivity against 15 other protein methyltransferases.
DC7927 EPZ011989 Featured EPZ011989 is a potent, orally-available EZH2 Inhibitor.
DC8012 EPZ015666 Featured EPZ015666 is a potent, selective and orally bioavailable PRMT5 inhibitor with Ki of 5 nM, >20,000-fold selectivity over other PMTs.
DC9267 EPZ015866 Featured EPZ015866(GSK591) is a potent, selective PRMT5 inhibitor.
DC26000 EPZ019997 Featured EPZ019997 is an orally active, reversible, and S-adenosyl-L-methionine (SAM) uncompetitive type I protein arginine methyltransferases (PRMTs) inhibitor (IC50=3.1 nM (PRMT1), 48 nM (PRMT3), 1148 nM (PRMT4), 5.7 nM (PRMT6), 1.7 nM (PRMT8)).
DC9822 EPZ020411 HCl Featured EPZ020411 is a potent and selective inhibitor of PRMT6 with IC50 of 10 nM, has ＞10 fold selectivity for PRMT6 over PRMT1 and PRMT8.
DC12529 EPZ020411 dihydrochloride EPZ020411 is a potent, selective PRMT6 inhibitor with IC50 of 10 nM, displays 10-fold and 20-fold selectivity over PRMT1/8, and >100-fold over other histone methyltransferases (PRMT3/4/5/7).
DC23134 EPZ020411 hydrochloride EPZ020411 is a potent, selective PRMT6 inhibitor with IC50 of 10 nM, displays 10-fold and 20-fold selectivity over PRMT1/8, and >100-fold over other histone methyltransferases (PRMT3/4/5/7).
DC20996 EPZ 025654 EPZ025654 (GSK 35336023) is a potent, selective arginine methyltransferase CARM1 inhibitor with IC50 of 3 nM.
DC22657 EPZ-030456 EPZ-030456 (EPZ030456) is a potent, selective SMYD3 inhibitor with biochem IC50 of 4 nM.
DC10887 EPZ031686 Featured EPZ031686 is a noncompetitive inhibitor for SMYD3 and MEKK2 with a Ki=1.2 and 1.1 nM respectively.
DC4242 Pinometostat(EPZ5676) Featured EPZ-5676 is a small molecule inhibitor of histone methyltransferase with potential antineoplastic activity.
DC7122 Tazemetostat(EPZ-6438) Featured EPZ-6438 is a potent, selective, and orally bioavailable small-molecule inhibitor of EZH2 enzymatic activity with Ki value of 2.5±0.5 nM.
DC8595 Equisetin Equisetin is an N-methylserine-derived acyl tetramic acid produced by a number of Fusarium species with antibiotic and cytotoxic activity.
DC20997 ER000444793 Featured ER-000444793 is a potent, cyclophilin D-independent inhibitor of mitochondrial permeability transition pore (mPTP) with with IC50 of 2.8 uM.
DC22468 ER-27319 maleate ER-27319 maleate is a potent, selective inhibitor of antigen or anti-IgE-mediated degranulation of rodent and human mast cells by selective inhibition of FcɛRI-mediated activation of Syk.
DC22090 ER-464195-01 ER-464195-01 is a specific, orally active inhibitor that inhibits Calreticulin (CRT) binding to integrin α subunits (ITGAs) with IC50 of 0.17, 0.36, and 0.23 uM in the interaction between CRT and ITGA α4, αL, and αM/α2/α5.
DC22433 ER-819762 ER-819762 is a novel potent, selective, orally active EP4 receptor antagonist with IC50 of 59 nM in cAMP-dependent reporter assay.
DC7410 Erastin Featured Erastin is a compound that interacts with VDAC, blocked and reversed mitochondrial depolarization after microtubule destabilizers in intact cells and antagonized tubulin-induced VDAC blockage in planar bilayers.
DC11238 ERD03 ERD03 (EXOSC3-RNA disrupting compound 3) is a small molecule EXOSC3-RNA disrupting (ERD) compound that binds specifically to EXOSC3 (Kd=17 uM), induces a PCH1B-like phenotype in zebrafish.

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