Home > Products > Novel inhibitors
Cat. No. Product name CAS No.
DC22846 NSC-34931

A anti-HIV-1 compound that interferes with HIV-I integrase binding to viral DNA..

6962-42-1
DC22455 Ro5-3335

A benzodiazepine inhibitor that directly interacts with RUNX1 and CBFβ, represses RUNX1/CBFβ-dependent transactivation in reporter assays.

30195-30-3
DC11768 TAM-16

A benzofuran class inhibitor of M. tuberculosis Pks13 (Polyketide Synthase 13).

2030241-59-7
DC22605 Benzophenonetetracarboxylic acid

A benzophenone tetracarboxylic derivative that can improve the activity and stability of alkaline phosphatases from psychrophilic and mesophilic organisms..

2479-49-4
DC20526 r(GGGGCC)n binder 1a

A bioactive, specific small molecule that targets RNA of the expanded repeat (r(GGGGCC)exp) with Kd of 9.7 uM.

70173-34-1
DC25030 Migrastatin

A biologically active natural product isolated from Streptomyces that has been shown to inhibit tumor cell migration.

314245-65-3
DC21819 WP760

A bis-anthracycline and melanoma selective agent that demonstrates anti-melanoma activity at low nanomolar concentrations.

DC22873 TM2 115 Featured

A BIX-01294 derivative that inhibit malaria parasite histone methyltransferases, resulting in rapid and irreversible parasite death.

1197196-47-6
DC7537 B-Raf inhibitor (BenzaMide)

A B-Raf inhibitor, pyrazine and pyrrolo[2,3-b]pyridine derivatives, useful in the treatment of cancer and proliferative diseases.

1315330-11-0
DC24040 AKT inhibitor

A broadly selective, potent, ATP-competitive Akt kinase inhibitor with IC50 of 0.5 nM(biochemical assay), and 0.31 nM (cell function assay).

1004990-28-6
DC23922 Cercosporamide Featured

A broad-spectrum natural antifungal compound that acts as a selective and highly potent fungal Pkc1 kinase inhibitor.

131436-22-1
DC23987 SU14813 maleate

A broad-spectrum RTKs inhibitor with IC50 ranging from 2 to 50 nM for VEGFR-1, VEGFR-2, PDGFRs, KIT, FLT3, and CSF1R/FMS.

849643-15-8
DC23920 GGTI298

A CAAZ peptidomimetic geranylgeranyltransferase I (GGTase I) inhibitor that inhibits the processing of geranylgeranylated Rap1A with little effect on processing of farnesylated Ha-Ras (IC50s are 3 and >10 uM respectively).

180977-44-0
DC22519 Norverapamil hydrochloride Featured

Norverapamil HCl is a calcium channel blocker. It is the main active metabolite of verapamil.

67812-42-4
DC24165 Aldicarb sulfone

A carbamate insecticide that acts as a fast-acting cholinesterase inhibitor..

1646-88-4
DC24166 Aldicarb

A carbamate insecticide that acts as a fast-acting cholinesterase inhibitor..

116-06-3
DC22369 Flumorph

A carboxylic acid amide (CAA) fungicide..

211867-47-9
DC22678 Acebutolol

A cardioselective beta blocker for the treatment of hypertension and arrhythmias..

37517-30-9
DC22489 Acebutolol hydrochloride Featured

Acebutolol HCl is a cardioselective beta-adrenergic antagonist with little effect on the bronchial receptors. The drug has stabilizing and quinidine-like effects on cardiac rhythm as well as weak inherent sympathomimetic action.

34381-68-5
DC22875 Hexamethylene bisacetamide

A cell differentiation inducer that inhibits activation of NF-κB function, Akt and ERK/MAPK cascade.

3073-59-4
DC11652 Ischemin sodium

A cell permeable CBP bromodomain inhibitor with Kd of 19 uM.

DC11653 Ischemin

A cell permeable CBP bromodomain inhibitor with Kd of 19 uM.

1357059-00-7
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